Synthesis of Borylated Hydrazino Acid Derivatives

نویسندگان

چکیده

Abstract α-Boryl-α-hydrazinoacetic acid is a highly functionalized boron-containing building block that can be easily accessed from readily available α-borylacetaldehyde. The hydrazine motif converted into variety of α-borylated azoles and diazines in straightforward protocol. Furthermore, the carboxy group derivatized to afford novel organoboron compounds should find applications various cross-coupling transformations.

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ژورنال

عنوان ژورنال: Synthesis

سال: 2021

ISSN: ['1791-5155', '1791-5856']

DOI: https://doi.org/10.1055/s-0040-1706046